| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM50391605 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_850392 (CHEMBL2150812) |
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| Ki | 0.808±n/a nM |
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| Citation |  Ida, Y; Matsubara, A; Nemoto, T; Saito, M; Hirayama, S; Fujii, H; Nagase, H Synthesis of quinolinomorphinan derivatives as highly selectived opioid receptor ligands. Bioorg Med Chem20:5810-31 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40577.25 |
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| Organism: | MOUSE |
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| Description: | P32300 |
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| Residue: | 372 |
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| Sequence: | MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTAC
TPSDGPGGGAAA
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| BDBM50391605 |
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| n/a |
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| Name | BDBM50391605 |
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| Synonyms: | CHEMBL2147918 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H26N2O3 |
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| Mol. Mass. | 402.4855 |
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| SMILES | COc1ccc2cc3C[C@@]4(O)[C@H]5Cc6ccc(O)cc6[C@@]4(CCN5C)Cc3nc2c1 |r,THB:24:23:9:19.13.12| |
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| Structure | 
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