| Reaction Details |
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 | Report a problem with these data |
| Target | Hydroxycarboxylic acid receptor 1 |
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| Ligand | BDBM50391815 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_850283 (CHEMBL2150703) |
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| EC50 | 129000±n/a nM |
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| Citation |  Dvorak, CA; Liu, C; Shelton, J; Kuei, C; Sutton, SW; Lovenberg, TW; Carruthers, NI Identification of Hydroxybenzoic Acids as Selective Lactate Receptor (GPR81) Agonists with Antilipolytic Effects. ACS Med Chem Lett3:637-639 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Hydroxycarboxylic acid receptor 1 |
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| Name: | Hydroxycarboxylic acid receptor 1 |
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| Synonyms: | G-protein coupled receptor 104 | GPR104 | GPR81 | HCA1 | HCAR1 | HCAR1_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 39313.04 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_850283 |
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| Residue: | 346 |
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| Sequence: | MYNGSCCRIEGDTISQVMPPLLIVAFVLGALGNGVALCGFCFHMKTWKPSTVYLFNLAVA
DFLLMICLPFRTDYYLRRRHWAFGDIPCRVGLFTLAMNRAGSIVFLTVVAADRYFKVVHP
HHAVNTISTRVAAGIVCTLWALVILGTVYLLLENHLCVQETAVSCESFIMESANGWHDIM
FQLEFFMPLGIILFCSFKIVWSLRRRQQLARQARMKKATRFIMVVAIVFITCYLPSVSAR
LYFLWTVPSSACDPSVHGALHITLSFTYMNSMLDPLVYYFSSPSFPKFYNKLKICSLKPK
QPGHSKTQRPEEMPISNLGRRSCISVANSFQSQSDGQWDPHIVEWH
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| BDBM50391815 |
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| n/a |
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| Name | BDBM50391815 |
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| Synonyms: | CHEMBL2146909 |
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| Type | Small organic molecule |
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| Emp. Form. | C7H5BrO3 |
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| Mol. Mass. | 217.017 |
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| SMILES | OC(=O)c1cc(O)cc(Br)c1 |
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| Structure | 
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