| Reaction Details |
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 | Report a problem with these data |
| Target | Matrilysin |
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| Ligand | BDBM50393207 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_850713 (CHEMBL2155982) |
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| Ki | >200±n/a nM |
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| Citation |  Mucha, A; Kafarski, P; Berlicki, L Remarkable potential of thea-aminophosphonate/phosphinate structural motif in medicinal chemistry. J Med Chem54:5955-80 (2011) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Matrilysin |
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| Name: | Matrilysin |
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| Synonyms: | MMP7 | MMP7_HUMAN | MPSL1 | Matrix metalloproteinase 7 | Matrix metalloproteinase-7 (MMP-7) | Matrix metalloproteinase-7 (MMP7) | PUMP1 |
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| Type: | Enzyme |
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| Mol. Mass.: | 29681.54 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P09237 |
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| Residue: | 267 |
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| Sequence: | MRLTVLCAVCLLPGSLALPLPQEAGGMSELQWEQAQDYLKRFYLYDSETKNANSLEAKLK
EMQKFFGLPITGMLNSRVIEIMQKPRCGVPDVAEYSLFPNSPKWTSKVVTYRIVSYTRDL
PHITVDRLVSKALNMWGKEIPLHFRKVVWGTADIMIGFARGAHGDSYPFDGPGNTLAHAF
APGTGLGGDAHFDEDERWTDGSSLGINFLYAATHELGHSLGMGHSSDPNAVMYPTYGNGD
PQNFKLSQDDIKGIQKLYGKRSNSRKK
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| BDBM50393207 |
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| n/a |
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| Name | BDBM50393207 |
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| Synonyms: | CHEMBL2153738 |
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| Type | Small organic molecule |
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| Emp. Form. | C37H36F3N4O7PS |
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| Mol. Mass. | 768.738 |
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| SMILES | NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@@H](CP(O)(=O)[C@H](Cc1ccccc1)NC(=O)OCc1ccccc1)Sc1ccccc1OC(F)(F)F |r| |
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| Structure | 
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