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TargetThromboxane A2 receptor
LigandBDBM50398348
Substrate/Competitorn/a
Meas. Tech.ChEMBL_875611 (CHEMBL2184409)
Ki 15±n/a nM
Citation Pease, JHoruk, R Chemokine receptor antagonists. J Med Chem55:9363-92 (2012) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Thromboxane A2 receptor
Name:Thromboxane A2 receptor
Synonyms:Prostanoid TP receptor | TA2R_HUMAN | TBXA2R | TXA2-R | Thromboxane | Thromboxane A2 receptor | Thromboxane Beta
Type:Enyzme
Mol. Mass.:37445.28
Organism:Homo sapiens (Human)
Description:P21731
Residue:343
Sequence:
MWPNGSSLGPCFRPTNITLEERRLIASPWFAASFCVVGLASNLLALSVLAGARQGGSHTR
SSFLTFLCGLVLTDFLGLLVTGTIVVSQHAALFEWHAVDPGCRLCRFMGVVMIFFGLSPL
LLGAAMASERYLGITRPFSRPAVASQRRAWATVGLVWAAALALGLLPLLGVGRYTVQYPG
SWCFLTLGAESGDVAFGLLFSMLGGLSVGLSFLLNTVSVATLCHVYHGQEAAQQRPRDSE
VEMMAQLLGIMVVASVCWLPLLVFIAQTVLRNPPAMSPAGQLSRTTEKELLIYLRVATWN
QILDPWVYILFRRAVLRRLQPRLSTRPRSLSLQPQLTQRSGLQ
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  Blast E-value cutoff:
BDBM50398348
n/a
NameBDBM50398348
Synonyms:CHEMBL2178581
TypeSmall organic molecule
Emp. Form.C25H20N2O3
Mol. Mass.396.4379
SMILESOC(=O)Cc1ccc2OCc3ccccc3\C(=C/Cn3cnc4ccccc34)c2c1
Structure
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