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TargetMu-type opioid receptor
LigandBDBM50398951
Substrate/Competitorn/a
Meas. Tech.ChEMBL_875495
Ki 0.2±n/a nM
Citation Moynihan HADerrick IBroadbear JHGreedy BMAceto MDHarris LSPurington LCThomas MPWoods JHTraynor JRHusbands SMLewis JW Fumaroylamino-4,5-epoxymorphinans and related opioids with irreversibleµ opioid receptor antagonist effects. J Med Chem 55:9868-74 (2012) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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  Blast E-value cutoff:
BDBM50398951
n/a
NameBDBM50398951
Synonyms:CHEMBL2179258
TypeSmall organic molecule
Emp. Form.C25H27NO7
Mol. Mass.453.4844
SMILESCOC(=O)\C=C\C(=O)O[C@]12CCC(=O)[C@@H]3Oc4c5c(C[C@H]1N(CC1CC1)CC[C@@]235)ccc4O |r|
Structure
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