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TargetMu-type opioid receptor
LigandBDBM50399639
Substrate/Competitorn/a
Meas. Tech.ChEMBL_878566 (CHEMBL2188651)
IC50 4.35±n/a nM
Citation Novoa, AVan Dorpe, SWynendaele, ESpetea, MBracke, NStalmans, SBetti, CChung, NNLemieux, CZuegg, JCooper, MATourwé, DDe Spiegeleer, BSchiller, PWBallet, S Variation of the net charge, lipophilicity, and side chain flexibility in Dmt(1)-DALDA: Effect on Opioid Activity and Biodistribution. J Med Chem55:9549-61 (2012) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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BDBM50399639
n/a
NameBDBM50399639
Synonyms:CHEMBL2181197
TypeSmall organic molecule
Emp. Form.C33H50N8O5
Mol. Mass.638.8007
SMILES[#6]-[#6]-[#6]-[#6]-[#6@H](-[#7](-[#6])-[#6](=O)-[#6@H](-[#6]-c1ccccc1)-[#7]-[#6](=O)-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#7]-[#6](=O)-[#6@@H](-[#7])-[#6]-c1c(-[#6])cc(-[#8])cc1-[#6])-[#6](-[#7])=O |r|
Structure
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