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TargetSigma non-opioid intracellular receptor 1
LigandBDBM50400741
Substrate/Competitorn/a
Meas. Tech.ChEMBL_880513
Ki 33±n/a nM
Citation Yu LFZhang HKGunosewoyo HKozikowski AP From a42 Nicotinic Ligands to the Discovery of s1 Receptor Ligands: Pharmacophore Analysis and Rational Design. ACS Med Chem Lett 3:1054-1058 (2012) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Sigma non-opioid intracellular receptor 1
Name:Sigma non-opioid intracellular receptor 1
Synonyms:Opioid receptor | Sigma | Sigma opioid receptor | Sigma-1
Type:Enzyme Catalytic Domain
Mol. Mass.:25266.54
Organism:RAT
Description:Q9R0C9
Residue:223
Sequence:
MPWAVGRRWAWITLFLTIVAVLIQAVWLWLGTQSFVFQREEIAQLARQYAGLDHELAFSR
LIVELRRLHPGHVLPDEELQWVFVNAGGWMGAMCLLHASLSEYVLLFGTALGSHGHSGRY
WAEISDTIISGTFHQWREGTTKSEVYYPGETVVHGPGEATAVEWGPNTWMVEYGRGVIPS
TLAFALSDTIFSTQDFLTLFYTLRAYARGLRLELTTYLFGQDP
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BDBM50400741
n/a
NameBDBM50400741
Synonyms:CHEMBL2165447
TypeSmall organic molecule
Emp. Form.C14H16N2O3
Mol. Mass.260.2884
SMILESC(Oc1cc(COc2ccccc2)on1)[C@@H]1CCN1 |r|
Structure
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