| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide FF receptor 1 |
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| Ligand | BDBM50402440 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_886542 (CHEMBL2215251) |
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| Ki | 29±n/a nM |
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| Citation |  Gealageas, R; Schneider, S; Humbert, JP; Bertin, I; Schmitt, M; Laboureyras, E; Dugave, C; Mollereau, C; Simonnet, G; Bourguignon, JJ; Simonin, F; Bihel, F Development of sub-nanomolar dipeptidic ligands of neuropeptide FF receptors. Bioorg Med Chem Lett22:7471-4 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Neuropeptide FF receptor 1 |
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| Name: | Neuropeptide FF receptor 1 |
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| Synonyms: | G-protein coupled receptor 147 | GPR147 | NPFF1 | NPFF1_HUMAN | NPFFR1 | RFamide-related peptide receptor OT7T022 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 47840.07 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1474637 |
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| Residue: | 430 |
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| Sequence: | MEGEPSQPPNSSWPLSQNGTNTEATPATNLTFSSYYQHTSPVAAMFIVAYALIFLLCMVG
NTLVCFIVLKNRHMHTVTNMFILNLAVSDLLVGIFCMPTTLVDNLITGWPFDNATCKMSG
LVQGMSVSASVFTLVAIAVERFRCIVHPFREKLTLRKALVTIAVIWALALLIMCPSAVTL
TVTREEHHFMVDARNRSYPLYSCWEAWPEKGMRRVYTTVLFSHIYLAPLALIVVMYARIA
RKLCQAPGPAPGGEEAADPRASRRRARVVHMLVMVALFFTLSWLPLWALLLLIDYGQLSA
PQLHLVTVYAFPFAHWLAFFNSSANPIIYGYFNENFRRGFQAAFRARLCPRPSGSHKEAY
SERPGGLLHRRVFVVVRPSDSGLPSESGPSSGAPRPGRLPLRNGRVAHHGLPREGPGCSH
LPLTIPAWDI
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| BDBM50402440 |
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| n/a |
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| Name | BDBM50402440 |
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| Synonyms: | CHEMBL2208305 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H38N6O3 |
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| Mol. Mass. | 482.6183 |
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| SMILES | [#7]\[#6](-[#7])=[#7]\[#6]-[#6]-[#6]-[#6@@H](-[#7]-[#6](=O)C12[#6]-[#6]-3-[#6]-[#6](-[#6]-[#6](-[#6]-3)-[#6]1)-[#6]2)-[#6](=O)-[#7]-[#6@@H](-[#6]-c1ccccc1)-[#6](-[#7])=O |r,TLB:9:11:14:18.17.16,THB:12:13:16:20.11.19,12:11:14.13.18:16,19:11:14:18.17.16,19:17:14:20.12.11| |
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| Structure | 
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