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TargetMu-type opioid receptor
LigandBDBM50240679
Substrate/Competitorn/a
Meas. Tech.ChEMBL_145305 (CHEMBL752840)
Ki 151±n/a nM
Citation Santagada, VBalboni, GCaliendo, GGuerrini, RSalvadori, SBianchi, CBryant, SDLazarus, LH Assessment of substitution in the second pharmacophore of Dmt-Tic analogues. Bioorg Med Chem Lett10:2745-8 (2000) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50240679
n/a
NameBDBM50240679
Synonyms:2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-1-(3-hydroxymethyl-3,4-dihydro-1H-isoquinolin-2-yl)-propan-1-one | 2-amino-3-(4-hydroxy-2,6-dimethylphenyl)-1-(3-hydroxymethyl-1,2,3,4-tetrahydro-2-isoquinolinyl)-(2S)-propan-1-one | CHEMBL328135
TypeSmall organic molecule
Emp. Form.C21H26N2O3
Mol. Mass.354.4427
SMILESCc1cc(O)cc(C)c1C[C@H](N)C(=O)N1Cc2ccccc2CC1CO
Structure
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