| Reaction Details |
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 | Report a problem with these data |
| Target | Aurora kinase A-interacting protein |
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| Ligand | BDBM50350908 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_502288 (CHEMBL983959) |
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| IC50 | 7943±n/a nM |
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| Citation |  Liddle, J; Bamborough, P; Barker, MD; Campos, S; Cousins, RP; Cutler, GJ; Hobbs, H; Holmes, DS; Ioannou, C; Mellor, GW; Morse, MA; Payne, JJ; Pritchard, JM; Smith, KJ; Tape, DT; Whitworth, C; Williamson, RA 4-Phenyl-7-azaindoles as potent and selective IKK2 inhibitors. Bioorg Med Chem Lett19:2504-8 (2009) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Aurora kinase A-interacting protein |
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| Name: | Aurora kinase A-interacting protein |
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| Synonyms: | AIP | AKIP | AKIP_HUMAN | AURKAIP1 | MRPS38 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 22379.19 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_502288 |
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| Residue: | 199 |
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| Sequence: | MLLGRLTSQLLRAVPWAGGRPPWPVSGVLGSRVCGPLYSTSPAGPGRAASLPRKGAQLEL
EEMLVPRKMSVSPLESWLTARCFLPRLDTGTAGTVAPPQSYQCPPSQIGEGAEQGDEGVA
DAPQIQCKNVLKIRRRKMNHHKYRKLVKKTRFLRRKVQEGRLRRKQIKFEKDLRRIWLKA
GLKEAPEGWQTPKIYLRGK
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| BDBM50350908 |
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| n/a |
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| Name | BDBM50350908 |
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| Synonyms: | CHEMBL520308 |
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| Type | Small organic molecule |
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| Emp. Form. | C17H19N3O3S |
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| Mol. Mass. | 345.416 |
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| SMILES | CN(CCO)S(=O)(=O)c1ccc(cc1)-c1ccnc2[nH]c(C)cc12 |
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| Structure | 
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