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TargetfMet-Leu-Phe receptor 1/2
LigandBDBM50418357
Substrate/Competitorn/a
Meas. Tech.ChEMBL_744724
IC50 2512±n/a nM
Citation Unitt JFagura MPhillips TKing SPerry MMorley AMacDonald CWeaver RChristie JBarber SMohammed RPaul MCook ABaxter A Discovery of small molecule human FPR1 receptor antagonists. Bioorg Med Chem Lett 21:2991-7 (2011) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
fMet-Leu-Phe receptor 1/2
Name:fMet-Leu-Phe receptor 1/2
Synonyms:Formyl peptide Receptor | formyl peptide receptor 1
Type:Enzyme Catalytic Domain
Mol. Mass.:38456.14
Organism:Homo sapiens (Human)
Description:gi_4503779
Residue:350
Sequence:
METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVT
TISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIA
LDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNF
SPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPL
RVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPML
YVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
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  Blast E-value cutoff:
BDBM50418357
n/a
NameBDBM50418357
Synonyms:CHEMBL1770304
TypeSmall organic molecule
Emp. Form.C21H23ClN2O3
Mol. Mass.386.872
SMILESOc1ccccc1C(=O)NC(C(=O)NC1CCCCC1)c1ccc(Cl)cc1
Structure
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