| Reaction Details |
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 | Report a problem with these data |
| Target | Solute carrier family 22 member 2 |
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| Ligand | BDBM50151860 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_838484 (CHEMBL2076055) |
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| IC50 | 5000±n/a nM |
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| Citation |  Urakami, Y; Okuda, M; Masuda, S; Akazawa, M; Saito, H; Inui, K Distinct characteristics of organic cation transporters, OCT1 and OCT2, in the basolateral membrane of renal tubules. Pharm Res18:1528-34 (2001) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Solute carrier family 22 member 2 |
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| Name: | Solute carrier family 22 member 2 |
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| Synonyms: | Adrenaline alpha2 | Oct2 | Organic cation transporter 2 | S22A2_RAT | Slc22a2 | Solute carrier family 22 member 2 | rOCT2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 62348.38 |
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| Organism: | RAT |
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| Description: | Adrenaline alpha2 0 RAT::Q9R0W2 |
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| Residue: | 555 |
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| Sequence: | MSTVDDILEHIGEFHLFQKQTFFLLALLSGAFTPIYVGIVFLGFTPDHHCWSPGAAKLSQ
RCGWSQAEELNYTVPGLGPSDEASFLSQCMRYEVDWNQSTLDCVDPLSSLAADRNQLPLG
PCEHGWVYNTPGSSIVTEFNLVCAHSWMLDLFQSVVNVGFFIGAMMIGYLADRFGRKFCL
LVTILINAISGALMAISPNYAWMLVFRFLQGLVSKAGWLIGYILITEFVGLGYRRMVGIC
YQIAFTVGLLILAGVAYVIPNWRWLQFAVTLPNFCFLLYFWCIPESPRWLISQNKIVKAM
KIIKHIAKKNGKSVPVSLQNLTPDEDAGKKLNPSFLDLVRTPQIRKHTLILMYNWFTSSV
LYQGLIMHMGLAGDNIYLDFFYSALVEFPAAFIIILTIDRVGRRYPWAVSNMVAGAACLA
SVFIPDDLQWLKITIACLGRMGITMAYEMVCLVNAELYPTYIRNLGVLVCSSMCDIGGII
TPFLVYRLTDIWMEFPLVVFAVVGLVAGALVLLLPETKGKALPETIEDAENMQRPRKKKE
KRIYLQVKQADRPLS
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| BDBM50151860 |
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| n/a |
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| Name | BDBM50151860 |
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| Synonyms: | 4-Acetylamino-N-(2-diethylamino-ethyl)-benzamide | ACECAINIDE | CHEMBL1097 | N-Acetyl Procainamide(<30%) | N-acetylprocainamide |
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| Type | Small organic molecule |
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| Emp. Form. | C15H23N3O2 |
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| Mol. Mass. | 277.362 |
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| SMILES | CCN(CC)CCNC(=O)c1ccc(NC(C)=O)cc1 |
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| Structure | 
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