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TargetSolute carrier family 22 member 1
LigandBDBM50029050
Substrate/Competitorn/a
Meas. Tech.ChEMBL_838514 (CHEMBL2078142)
Ki 1600000±n/a nM
Citation Urakami, Y; Okuda, M; Masuda, S; Akazawa, M; Saito, H; Inui, K Distinct characteristics of organic cation transporters, OCT1 and OCT2, in the basolateral membrane of renal tubules. Pharm Res18:1528-34 (2001) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Solute carrier family 22 member 1
Name:Solute carrier family 22 member 1
Synonyms:Adrenaline alpha1 | Oct1 | Organic cation transporter 1 | S22A1_RAT | Slc22a1 | Solute carrier family 22 member 1 | adrenergic Alpha1 | rOCT1
Type:Enzyme Catalytic Domain
Mol. Mass.:61538.40
Organism:RAT
Description:Adrenaline alpha1 0 RAT::Q63089
Residue:556
Sequence:
MPTVDDVLEQVGEFGWFQKQAFLLLCLISASLAPIYVGIVFLGFTPGHYCQNPGVAELSQ
RCGWSQAEELNYTVPGLGPSDEASFLSQCMRYEVDWNQSTLDCVDPLSSLVANRSQLPLG
PCEHGWVYDTPGSSIVTEFNLVCGDAWKVDLFQSCVNLGFFLGSLVVGYIADRFGRKLCL
LVTTLVTSVSGVLTAVAPDYTSMLLFRLLQGMVSKGSWVSGYTLITEFVGSGYRRTTAIL
YQMAFTVGLVGLAGVAYAIPDWRWLQLAVSLPTFLFLLYYWFVPESPRWLLSQKRTTRAV
RIMEQIAQKNGKVPPADLKMLCLEEDASEKRSPSFADLFRTPNLRKHTVILMYLWFSCAV
LYQGLIMHVGATGANLYLDFFYSSLVEFPAAFIILVTIDRIGRIYPIAASNLVTGAACLL
MIFIPHELHWLNVTLACLGRMGATIVLQMVCLVNAELYPTFIRNLGMMVCSALCDLGGIF
TPFMVFRLMEVWQALPLILFGVLGLTAGAMTLLLPETKGVALPETIEEAENLGRRKSKAK
ENTIYLQVQTGKSSST
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  Blast E-value cutoff:
BDBM50029050
n/a
NameBDBM50029050
Synonyms:(-)-(R)-epinephrine | (-)-3,4-dihydroxy-alpha-((methylamino)methyl)benzyl alcohol | (-)-adrenaline | (R)-(-)-adrenaline | (R)-adrenaline | 4-[(1R)-1-hydroxy-2-(methylamino)ethyl]benzene-1,2-diol | Adrenalin | CHEMBL679 | EPINEPHRINE | adrenaline | levoepinephrine
TypeSmall organic molecule
Emp. Form.C9H13NO3
Mol. Mass.183.2044
SMILESCNC[C@H](O)c1ccc(O)c(O)c1 |r|
Structure
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