| Reaction Details |
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 | Report a problem with these data |
| Target | Solute carrier organic anion transporter family member 1A3 |
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| Ligand | BDBM50390979 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_838743 (CHEMBL2078569) |
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| Ki | 21000±n/a nM |
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| Citation |  Takeuchi, A; Masuda, S; Saito, H; Hashimoto, Y; Inui, K Trans-stimulation effects of folic acid derivatives on methotrexate transport by rat renal organic anion transporter, OAT-K1. J Pharmacol Exp Ther293:1034-9 (2000) [PubMed] |
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| More Info.: | Get all data from this article, Assay Method |
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| Solute carrier organic anion transporter family member 1A3 |
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| Name: | Solute carrier organic anion transporter family member 1A3 |
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| Synonyms: | OAT-K1 | OAT-K2 | Oatp1a3 | SO1A3_RAT | Slc21a4 | Slco1a3 | Sodium-independent organic anion transporter K1 | Solute carrier family 21 member 4 | rOAT-K |
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| Type: | PROTEIN |
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| Mol. Mass.: | 73829.31 |
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| Organism: | Rattus norvegicus |
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| Description: | ChEMBL_838743 |
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| Residue: | 670 |
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| Sequence: | MGDLEKGAATHGAGCFAKIKVFLMALTCAYVSKSLSGTFMSSMLTQIERQFGIPTAIVGF
INGSFEIGNLLLIIFVSYFGMKLHRPIVIGVGCAVMGLGCFIISLPHFLMGRYEYETTIL
PTSNLSSNSFLCMENQTQTLNPAQDPAECVKEVKSLMWIYVLVGNIIRGIGETPIMPLGV
SYIENFAKSENSPLYIGILETGKMIGPIFGLLLGSFCASIYVDTGSVNTDDLTITPTDIR
WVGAWWIGFLVCAGVNILISIPFFFFPKTLPKEGLQENVDGTENAKEESTEKRPRKKNRG
ITKDFFPFLKSPVLQPDLHAVHPYKVLQVNAFNIYFSFLPKYLENQYGKSTAEVIFLMGV
YNLPAICIGYLIAGFMMKKFKITVKTAAFLAFCLSLSEYSFGFCNFLITCDNVPVAGLTN
SYERDQKPLYLENNVLADCNTRCSCLTKTWDPVCGDNGLAYMSACLAGCEKSVGTGTNMV
FHNCSCIQSPGNSSAVLGLCNKGPECTNKLQYLLILSGFLSILYSFAAIPGYMVFLRCIK
SEEKSLGIGIHAFCIRVFAGIPAPIYFGALIDRTCLHWGTQKCGAPGACRMYDINSFRRI
YLGMSAALRGSSYLPAFVIVILTRKFSLPGKINSSEMEIAEMKLTEKESQCTDVHRNPKF
KNDGELKTKL
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| BDBM50390979 |
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| n/a |
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| Name | BDBM50390979 |
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| Synonyms: | BROMOSULFOPHTHALEIN |
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| Type | Small organic molecule |
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| Emp. Form. | C20H8Br4O10S2 |
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| Mol. Mass. | 792.019 |
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| SMILES | Oc1ccc(cc1S([O-])(=O)=O)C1(OC(=O)c2c1c(Br)c(Br)c(Br)c2Br)c1ccc(O)c(c1)S([O-])(=O)=O |
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| Structure | 
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