| Reaction Details |
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 | Report a problem with these data |
| Target | Solute carrier family 22 member 3 |
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| Ligand | BDBM39687 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_839283 (CHEMBL2077954) |
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| IC50 | 90±n/a nM |
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| Citation |  Hayer-Zillgen, M; Brüss, M; Bönisch, H Expression and pharmacological profile of the human organic cation transporters hOCT1, hOCT2 and hOCT3. Br J Pharmacol136:829-36 (2002) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Solute carrier family 22 member 3 |
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| Name: | Solute carrier family 22 member 3 |
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| Synonyms: | EMT | EMTH | Extraneuronal monoamine transporter | OCT3 | Organic cation transporter 3 | S22A3_HUMAN | SLC22A3 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 61292.57 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_934315 |
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| Residue: | 556 |
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| Sequence: | MPSFDEALQRVGEFGRFQRRVFLLLCLTGVTFAFLFVGVVFLGTQPDHYWCRGPSAAALA
ERCGWSPEEEWNRTAPASRGPEPPERRGRCQRYLLEAANDSASATSALSCADPLAAFPNR
SAPLVPCRGGWRYAQAHSTIVSEFDLVCVNAWMLDLTQAILNLGFLTGAFTLGYAADRYG
RIVIYLLSCLGVGVTGVVVAFAPNFPVFVIFRFLQGVFGKGTWMTCYVIVTEIVGSKQRR
IVGIVIQMFFTLGIIILPGIAYFIPNWQGIQLAITLPSFLFLLYYWVVPESPRWLITRKK
GDKALQILRRIAKCNGKYLSSNYSEITVTDEEVSNPSFLDLVRTPQMRKCTLILMFAWFT
SAVVYQGLVMRLGIIGGNLYIDFFISGVVELPGALLILLTIERLGRRLPFAASNIVAGVA
CLVTAFLPEGIAWLRTTVATLGRLGITMAFEIVYLVNSELYPTTLRNFGVSLCSGLCDFG
GIIAPFLLFRLAAVWLELPLIIFGILASICGGLVMLLPETKGIALPETVDDVEKLGSPHS
CKCGRNKKTPVSRSHL
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| BDBM39687 |
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| n/a |
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| Name | BDBM39687 |
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| Synonyms: | (2E)-1-ethyl-2-[(1-ethyl-2-quinolin-1-iumyl)methylidene]quinoline;chloride | (2E)-1-ethyl-2-[(1-ethylquinolin-1-ium-2-yl)methylene]quinoline;chloride | (2E)-1-ethyl-2-[(1-ethylquinolin-1-ium-2-yl)methylidene]quinoline;chloride | 1-ethyl-2-[(1-ethyl-2(1H)-quinolinylidene)methyl]quinolinium chloride | CHEMBL1197556 | MLS000532635 | SMR000137574 | cid_5717105 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H23N2 |
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| Mol. Mass. | 327.4416 |
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| SMILES | CCN1\C(=C\c2ccc3ccccc3[n+]2CC)C=Cc2ccccc12 |c:19| |
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| Structure | 
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