| Reaction Details |
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 | Report a problem with these data |
| Target | Solute carrier family 22 member 3 |
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| Ligand | BDBM50017679 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_839283 (CHEMBL2077954) |
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| IC50 | 6130±n/a nM |
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| Citation |  Hayer-Zillgen, M; Brüss, M; Bönisch, H Expression and pharmacological profile of the human organic cation transporters hOCT1, hOCT2 and hOCT3. Br J Pharmacol136:829-36 (2002) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Solute carrier family 22 member 3 |
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| Name: | Solute carrier family 22 member 3 |
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| Synonyms: | EMT | EMTH | Extraneuronal monoamine transporter | OCT3 | Organic cation transporter 3 | S22A3_HUMAN | SLC22A3 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 61292.57 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_934315 |
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| Residue: | 556 |
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| Sequence: | MPSFDEALQRVGEFGRFQRRVFLLLCLTGVTFAFLFVGVVFLGTQPDHYWCRGPSAAALA
ERCGWSPEEEWNRTAPASRGPEPPERRGRCQRYLLEAANDSASATSALSCADPLAAFPNR
SAPLVPCRGGWRYAQAHSTIVSEFDLVCVNAWMLDLTQAILNLGFLTGAFTLGYAADRYG
RIVIYLLSCLGVGVTGVVVAFAPNFPVFVIFRFLQGVFGKGTWMTCYVIVTEIVGSKQRR
IVGIVIQMFFTLGIIILPGIAYFIPNWQGIQLAITLPSFLFLLYYWVVPESPRWLITRKK
GDKALQILRRIAKCNGKYLSSNYSEITVTDEEVSNPSFLDLVRTPQMRKCTLILMFAWFT
SAVVYQGLVMRLGIIGGNLYIDFFISGVVELPGALLILLTIERLGRRLPFAASNIVAGVA
CLVTAFLPEGIAWLRTTVATLGRLGITMAFEIVYLVNSELYPTTLRNFGVSLCSGLCDFG
GIIAPFLLFRLAAVWLELPLIIFGILASICGGLVMLLPETKGIALPETVDDVEKLGSPHS
CKCGRNKKTPVSRSHL
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| BDBM50017679 |
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| n/a |
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| Name | BDBM50017679 |
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| Synonyms: | Benzyl-(2-chloro-ethyl)-(1-methyl-2-phenoxy-ethyl)-amine | CHEMBL753 | Dibenzyline | PHENOXYBENZAMINE |
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| Type | Small organic molecule |
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| Emp. Form. | C18H22ClNO |
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| Mol. Mass. | 303.826 |
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| SMILES | CC(COc1ccccc1)N(CCCl)Cc1ccccc1 |
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| Structure | 
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