| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM50424108 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_937282 (CHEMBL2318811) |
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| Ki | >1000±n/a nM |
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| Citation |  Nemoto, T; Yamamoto, N; Wada, N; Harada, Y; Tomatsu, M; Ishihara, M; Hirayama, S; Iwai, T; Fujii, H; Nagase, H The effect of 17-N substituents on the activity of the opioid¿ receptor in nalfurafine derivatives. Bioorg Med Chem Lett23:268-72 (2012) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40577.25 |
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| Organism: | MOUSE |
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| Description: | P32300 |
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| Residue: | 372 |
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| Sequence: | MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTAC
TPSDGPGGGAAA
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| BDBM50424108 |
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| n/a |
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| Name | BDBM50424108 |
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| Synonyms: | CHEMBL2315357 |
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| Type | Small organic molecule |
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| Emp. Form. | C25H30F2N2O5 |
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| Mol. Mass. | 476.5129 |
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| SMILES | CN(CCC[C@@]1(O)[C@H]2Cc3ccc(O)c(O)c3[C@@H]1CCN2CC(F)F)C(=O)\C=C\c1ccoc1 |r| |
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| Structure | 
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