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TargetMu-type opioid receptor
LigandBDBM50268462
Substrate/Competitorn/a
Meas. Tech.ChEMBL_940036 (CHEMBL2327845)
IC50 260±n/a nM
Citation Carroll, FICarlezon, WA Development of¿ opioid receptor antagonists. J Med Chem56:2178-95 (2013) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Mu-type opioid receptor
Name:Mu-type opioid receptor
Synonyms:M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:Enzyme Catalytic Domain
Mol. Mass.:11165.58
Organism:GUINEA PIG
Description:P97266
Residue:98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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BDBM50268462
n/a
NameBDBM50268462
Synonyms:CHEMBL506616 | c[L-Phe-D-pro-L-Phe-L-trp]
TypeSmall organic molecule
Emp. Form.C34H35N5O4
Mol. Mass.577.6728
SMILESO=C1N[C@@H](Cc2ccccc2)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](Cc2ccccc2)C(=O)N2CCC[C@H]12 |r|
Structure
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