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TargetCAMK2A
LigandBDBM50430016
Substrate/Competitorn/a
Meas. Tech.ChEMBL_946301
IC50 30±n/a nM
Citation Gomez-Monterrey ISala MRusciano MRMonaco SMaione ASIaccarino GTortorella PD'Ursi AMScrima MCarotenuto ADe Rosa GBertamino AVernieri EGrieco PNovellino EIllario MCampiglia P Characterization of a selective CaMKII peptide inhibitor. Eur J Med Chem 62:425-34 (2013) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
CAMK2A
Name:CAMK2A
Synonyms:CaM kinase II | CaM kinase II alpha | Calcium/calmodulin-dependent protein kinase type II subunit alpha (CAMK2a)
Type:Enzyme Catalytic Domain
Mol. Mass.:54093.63
Organism:Homo sapiens (Human)
Description:gi_25952118
Residue:478
Sequence:
MATITCTRFTEEYQLFEELGKGAFSVVRRCVKVLAGQEYAAKIINTKKLSARDHQKLERE
ARICRLLKHPNIVRLHDSISEEGHHYLIFDLVTGGELFEDIVAREYYSEADASHCIQQIL
EAVLHCHQMGVVHRDLKPENLLLASKLKGAAVKLADFGLAIEVEGEQQAWFGFAGTPGYL
SPEVLRKDPYGKPVDLWACGVILYILLVGYPPFWDEDQHRLYQQIKAGAYDFPSPEWDTV
TPEAKDLINKMLTINPSKRITAAEALKHPWISHRSTVASCMHRQETVDCLKKFNARRKLK
GAILTTMLATRNFSGGKSGGNKKSDGVKESSESTNTTIEDEDTKVRKQEIIKVTEQLIEA
ISNGDFESYTKMCDPGMTAFEPEALGNLVEGLDFHRFYFENLWSRNSKPVHTTILNPHIH
LMGDESACIAYIRITQYLDAGGIPRTAQSEETRVWHRRDGKWQIVHFHRSGAPSVLPH
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50430016
n/a
NameBDBM50430016
Synonyms:CHEMBL2335444
TypeSmall organic molecule
Emp. Form.C197H335N67O41S2
Mol. Mass.4362.322
SMILESn/a
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: