| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50430627 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_948260 (CHEMBL2340178) |
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| Ki | 2.7±n/a nM |
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| Citation |  Greedy, BM; Bradbury, F; Thomas, MP; Grivas, K; Cami-Kobeci, G; Archambeau, A; Bosse, K; Clark, MJ; Aceto, M; Lewis, JW; Traynor, JR; Husbands, SM Orvinols with mixed kappa/mu opioid receptor agonist activity. J Med Chem56:3207-16 (2013) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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| BDBM50430627 |
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| n/a |
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| Name | BDBM50430627 |
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| Synonyms: | CHEMBL2338736 |
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| Type | Small organic molecule |
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| Emp. Form. | C30H43NO4 |
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| Mol. Mass. | 481.6667 |
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| SMILES | CCCCC[C@](C)(O)[C@H]1C[C@]23CC[C@]1(OC)[C@@H]1Oc4c5c(C[C@H]2N(CC2CC2)CC[C@@]315)ccc4O |r,THB:5:8:30.16:11.12| |
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| Structure | 
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