| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50430799 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_943433 (CHEMBL2341877) |
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| IC50 | 0.467000±n/a nM |
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| Citation |  Liu, X; Wang, Y; Xing, Y; Yu, J; Ji, H; Kai, M; Wang, Z; Wang, D; Zhang, Y; Zhao, D; Wang, R Design, synthesis, and pharmacological characterization of novel endomorphin-1 analogues as extremely potentµ-opioid agonists. J Med Chem56:3102-14 (2013) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 11165.58 |
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| Organism: | GUINEA PIG |
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| Description: | P97266 |
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| Residue: | 98 |
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| Sequence: | YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSI
FTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
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|
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| BDBM50430799 |
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| n/a |
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| Name | BDBM50430799 |
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| Synonyms: | CHEMBL2334772 |
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| Type | Small organic molecule |
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| Emp. Form. | C37H41N5O6 |
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| Mol. Mass. | 651.7513 |
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| SMILES | Cc1cc(O)cc(C)c1C[C@H](N)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(=O)N[C@H](C(=C)C(O)=O)c1ccccc1 |r| |
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| Structure | 
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