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TargetCasein kinase I isoform alpha
LigandBDBM50432006
Substrate/Competitorn/a
Meas. Tech.ChEMBL_954191 (CHEMBL2351706)
IC50>10000±n/a nM
Citation Elagawany, MIbrahim, MAAli Ahmed, HEEl-Etrawy, AShGhiaty, AAbdel-Samii, ZKEl-Feky, SABajorath, J Design, synthesis, and molecular modelling of pyridazinone and phthalazinone derivatives as protein kinases inhibitors. Bioorg Med Chem Lett23:2007-13 (2013) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Casein kinase I isoform alpha
Name:Casein kinase I isoform alpha
Synonyms:CK1 | CKI-alpha | CSNK1A1 | KC1A_PIG
Type:PROTEIN
Mol. Mass.:14639.55
Organism:Sus scrofa
Description:ChEMBL_939731
Residue:125
Sequence:
GEEVAVKLESQKARHPQLLYESKLYKILQGGVGIPHIRWYGQEKDYNVLVMDLLGPSLED
LFNFCSRRFTMKTVLMLADQMISRIEYVHTKNFIHRDIKPDNFLMGIGRHCNKLFLIDFG
LAKKY
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BDBM50432006
n/a
NameBDBM50432006
Synonyms:CHEMBL2348737
TypeSmall organic molecule
Emp. Form.C17H13N3O2
Mol. Mass.291.304
SMILESO=C(Nc1cc(-c2ccccc2)c(=O)[nH]n1)c1ccccc1
Structure
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