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TargetCasein kinase I isoform alpha
LigandBDBM50431993
Substrate/Competitorn/a
Meas. Tech.ChEMBL_954191 (CHEMBL2351706)
IC50>10000±n/a nM
Citation Elagawany, MIbrahim, MAAli Ahmed, HEEl-Etrawy, AShGhiaty, AAbdel-Samii, ZKEl-Feky, SABajorath, J Design, synthesis, and molecular modelling of pyridazinone and phthalazinone derivatives as protein kinases inhibitors. Bioorg Med Chem Lett23:2007-13 (2013) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Casein kinase I isoform alpha
Name:Casein kinase I isoform alpha
Synonyms:CK1 | CKI-alpha | CSNK1A1 | KC1A_PIG
Type:PROTEIN
Mol. Mass.:14639.55
Organism:Sus scrofa
Description:ChEMBL_939731
Residue:125
Sequence:
GEEVAVKLESQKARHPQLLYESKLYKILQGGVGIPHIRWYGQEKDYNVLVMDLLGPSLED
LFNFCSRRFTMKTVLMLADQMISRIEYVHTKNFIHRDIKPDNFLMGIGRHCNKLFLIDFG
LAKKY
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BDBM50431993
n/a
NameBDBM50431993
Synonyms:CHEMBL2348747
TypeSmall organic molecule
Emp. Form.C17H15N3O
Mol. Mass.277.3205
SMILESO=c1cc(c(NCc2ccccc2)n[nH]1)-c1ccccc1
Structure
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