| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 55 |
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| Ligand | BDBM50398218 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_963381 (CHEMBL2388878) |
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| IC50 | 113±n/a nM |
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| Citation |  Rempel, V; Volz, N; Gläser, F; Nieger, M; Bräse, S; Müller, CE Antagonists for the orphan G-protein-coupled receptor GPR55 based on a coumarin scaffold. J Med Chem56:4798-810 (2013) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| G-protein coupled receptor 55 |
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| Name: | G-protein coupled receptor 55 |
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| Synonyms: | G protein-coupled receptor 55 | GPR55 | GPR55_HUMAN |
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| Type: | PROTEIN |
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| Mol. Mass.: | 36649.72 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1292265 |
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| Residue: | 319 |
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| Sequence: | MSQQNTSGDCLFDGVNELMKTLQFAVHIPTFVLGLLLNLLAIHGFSTFLKNRWPDYAATS
IYMINLAVFDLLLVLSLPFKMVLSQVQSPFPSLCTLVECLYFVSMYGSVFTICFISMDRF
LAIRYPLLVSHLRSPRKIFGICCTIWVLVWTGSIPIYSFHGKVEKYMCFHNMSDDTWSAK
VFFPLEVFGFLLPMGIMGFCCSRSIHILLGRRDHTQDWVQQKACIYSIAASLAVFVVSFL
PVHLGFFLQFLVRNSFIVECRAKQSISFFLQLSMCFSNVNCCLDVFCYYFVIKEFRMNIR
AHRPSRVQLVLQDTTISRG
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| BDBM50398218 |
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| n/a |
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| Name | BDBM50398218 |
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| Synonyms: | CHEMBL2181542 |
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| Type | Small organic molecule |
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| Emp. Form. | C26H32O4 |
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| Mol. Mass. | 408.5299 |
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| SMILES | CCCCCCCC(C)(C)c1cc(O)c2cc(Cc3ccccc3O)c(=O)oc2c1 |
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| Structure | 
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