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TargetG-protein coupled receptor 35
LigandBDBM50436011
Substrate/Competitorn/a
Meas. Tech.ChEMBL_964304
EC50 128±n/a nM
Citation Funke MThimm DSchiedel ACMüller CE 8-Benzamidochromen-4-one-2-carboxylic acids: potent and selective agonists for the orphan G protein-coupled receptor GPR35. J Med Chem 56:5182-97 (2013) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
G-protein coupled receptor 35
Name:G-protein coupled receptor 35
Synonyms:G protein-coupled receptor 35
Type:Enzyme Catalytic Domain
Mol. Mass.:34085.57
Organism:Homo sapiens (Human)
Description:gi_33695097
Residue:309
Sequence:
MNGTYNTCGSSDLTWPPAIKLGFYAYLGVLLVLGLLLNSLALWVFCCRMQQWTETRIYMT
NLAVADLCLLCTLPFVLHSLRDTSDTPLCQLSQGIYLTNRYMSISLVTAIAVDRYVAVRH
PLRARGLRSPRQAAAVCAVLWVLVIGSLVARWLLGIQEGGFCFRSTRHNFNSMAFPLLGF
YLPLAVVVFCSLKVVTALAQRPPTDVGQAEATRKAARMVWANLLVFVVCFLPLHVGLTVR
LAVGWNACALLETIRRALYITSKLSDANCCLDAICYYYMAKEFQEASALAVAPSAKAHKS
QDSLCVTLA
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  Blast E-value cutoff:
BDBM50436011
n/a
NameBDBM50436011
Synonyms:CHEMBL2392178
TypeSmall organic molecule
Emp. Form.C18H10BrNO7
Mol. Mass.432.179
SMILESOC(=O)c1cc(=O)c2cc(Br)cc(NC(=O)c3ccc4OCOc4c3)c2o1
Structure
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