| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 35 |
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| Ligand | BDBM50436009 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_964310 (CHEMBL2395572) |
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| EC50 | 5030±n/a nM |
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| Citation |  Funke, M; Thimm, D; Schiedel, AC; Müller, CE 8-Benzamidochromen-4-one-2-carboxylic acids: potent and selective agonists for the orphan G protein-coupled receptor GPR35. J Med Chem56:5182-97 (2013) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| G-protein coupled receptor 35 |
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| Name: | G-protein coupled receptor 35 |
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| Synonyms: | GPR35_MOUSE | Gpr35 | KYNA receptor | Kynurenic acid receptor |
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| Type: | PROTEIN |
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| Mol. Mass.: | 34163.11 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_107606 |
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| Residue: | 307 |
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| Sequence: | MNSTTCNSTLTWPASVNNFFIIYSALLLVLGLLLNSVALWVFCYRMHQWTETRIYMTNLA
VADLCLLCSLPFVLYSLKYSSSDTPVCQLSQGIYLANRYMSISLVTAIAVDRYVAVRHPL
RARELRSPRQAAAVCVALWVIVVTSLVVRWRLGMQEGGFCFSSQTRRNFSTTAFSLLGFY
LPLAIVVFCSLQVVTVLSRRPAADVGQAEATQKATHMVWANLAVFVICFLPLHVVLTVQV
SLNLNTCAARDTFSRALSITGKLSDTNCCLDAICYYYMAREFQEASKPATSSNTPHKSQD
SQILSLT
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| BDBM50436009 |
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| n/a |
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| Name | BDBM50436009 |
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| Synonyms: | CHEMBL2392157 |
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| Type | Small organic molecule |
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| Emp. Form. | C18H13NO6 |
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| Mol. Mass. | 339.2989 |
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| SMILES | COc1ccc(cc1)C(=O)Nc1cccc2c1oc(cc2=O)C(O)=O |
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| Structure | 
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