| Reaction Details |
|---|
 | Report a problem with these data |
| Target | G-protein coupled receptor 35 |
|---|
| Ligand | BDBM35525 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_983067 (CHEMBL2427427) |
|---|
| EC50 | 1300±n/a nM |
|---|
| Citation |  Thimm, D; Funke, M; Meyer, A; Müller, CE 6-Bromo-8-(4-[(3)H]methoxybenzamido)-4-oxo-4H-chromene-2-carboxylic Acid: a powerful tool for studying orphan G protein-coupled receptor GPR35. J Med Chem56:7084-99 (2013) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| G-protein coupled receptor 35 |
|---|
| Name: | G-protein coupled receptor 35 |
|---|
| Synonyms: | G protein-coupled receptor 35 | GPR35 | GPR35_HUMAN |
|---|
| Type: | Enzyme Catalytic Domain |
|---|
| Mol. Mass.: | 34085.57 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | gi_33695097 |
|---|
| Residue: | 309 |
|---|
| Sequence: | MNGTYNTCGSSDLTWPPAIKLGFYAYLGVLLVLGLLLNSLALWVFCCRMQQWTETRIYMT
NLAVADLCLLCTLPFVLHSLRDTSDTPLCQLSQGIYLTNRYMSISLVTAIAVDRYVAVRH
PLRARGLRSPRQAAAVCAVLWVLVIGSLVARWLLGIQEGGFCFRSTRHNFNSMAFPLLGF
YLPLAVVVFCSLKVVTALAQRPPTDVGQAEATRKAARMVWANLLVFVVCFLPLHVGLTVR
LAVGWNACALLETIRRALYITSKLSDANCCLDAICYYYMAKEFQEASALAVAPSAKAHKS
QDSLCVTLA
|
|
|
|---|
| BDBM35525 |
|---|
| n/a |
|---|
| Name | BDBM35525 |
|---|
| Synonyms: | 3,3''''-methylenebis(4-hydroxy-coumarin | 3,3''''-methylenebis(4-hydroxycoumarin) | 3,3''''-methylenebis[4-hydroxycoumarin | 4-hydroxy-3-((4-hydroxy-2-oxo-2H-chromen-3-yl)methyl)-2H-chromen-2-one | Bishydroxycoumarin | CHEMBL1466 | DICUMAROL | dicoumarol | symmetric dicoumarol analogue, 1 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C19H12O6 |
|---|
| Mol. Mass. | 336.295 |
|---|
| SMILES | Oc1c(Cc2c(O)c3ccccc3oc2=O)c(=O)oc2ccccc12 |
|---|
| Structure | 
|
|---|
Search and Browse
