| Reaction Details |
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 | Report a problem with these data |
| Target | Proteinase-activated receptor 2 |
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| Ligand | BDBM50440870 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_984148 (CHEMBL2432076) |
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| IC50 | 50000±n/a nM |
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| Citation |  Yau, MK; Liu, L; Fairlie, DP Toward drugs for protease-activated receptor 2 (PAR2). J Med Chem56:7477-97 (2013) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Proteinase-activated receptor 2 |
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| Name: | Proteinase-activated receptor 2 |
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| Synonyms: | F2rl1 | PAR2_RAT | Par2 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 44466.34 |
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| Organism: | RAT |
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| Description: | PAR2 F2RL1 RAT::Q63645 |
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| Residue: | 397 |
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| Sequence: | MRSLSLAWLLGGITLLAASASCNRTVNAPGPNSKGRSLIGRLDTPPPITGKGAPVEPGFS
VDEFSASVLTGKLTTVFLPVIYIIVFVIGLPSNGMALWVFFFRTKKKHPAVIYMANLALA
DLLSVIWFPLKISYHLHGNDWTYGDALCKVLIGFFYGNMYCSILFMTCLSVQRYWVIVNP
MGHSRKRANIAVGVSLAIWLLIFLVTIPLYVMRQTIYIPALNITTCHDVLPEEVLVGDMF
SYFLSLAIGVFLFPALLTASAYVLMIKTLRSSAMDEHSEKKRRRAIRLIITVLSMYFICF
APSNVLLVVHYFLIKSQRQSHVYALYLVALCLSTLNSCIDPFVYYFVSKDFRDQARNALL
CRSVRTVKRMQISLTSNKFSRKSSSYSSSSTSVKTSY
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| BDBM50440870 |
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| n/a |
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| Name | BDBM50440870 |
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| Synonyms: | CHEMBL2431726 |
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| Type | Small organic molecule |
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| Emp. Form. | C29H56N10O7 |
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| Mol. Mass. | 656.8177 |
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| SMILES | [#6]-[#6]-[#6@H](-[#6])-[#6@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#8])-[#7]-[#6](=O)-[#6@@H](-[#7])-[#6]-[#6](-[#6])-[#6])-[#6](=O)-[#7]-[#6]-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6](-[#6])-[#6])-[#6](-[#7])=O |r| |
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| Structure | 
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