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TargetNeuropeptide Y receptor type 4
LigandBDBM50197025
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1282126 (CHEMBL3102010)
EC50 141±n/a nM
Citation Albertsen, LAndersen, JJPaulsson, JFThomsen, JKNorrild, JCStrømgaard, K Design and Synthesis of Peptide YY Analogues with C-terminal Backbone Amide-to-Ester Modifications. ACS Med Chem Lett4:1228-32 (2013) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Neuropeptide Y receptor type 4
Name:Neuropeptide Y receptor type 4
Synonyms:NPY-Y4 | NPY4-R | NPY4R | NPY4R_HUMAN | PP1 | PPYR1 | Pancreatic polypeptide receptor 1
Type:Enzyme Catalytic Domain
Mol. Mass.:42207.58
Organism:Homo sapiens (Human)
Description:NPY-Y4 PPYR1 HUMAN::P50391
Residue:375
Sequence:
MNTSHLLALLLPKSPQGENRSKPLGTPYNFSEHCQDSVDVMVFIVTSYSIETVVGVLGNL
CLMCVTVRQKEKANVTNLLIANLAFSDFLMCLLCQPLTAVYTIMDYWIFGETLCKMSAFI
QCMSVTVSILSLVLVALERHQLIINPTGWKPSISQAYLGIVLIWVIACVLSLPFLANSIL
ENVFHKNHSKALEFLADKVVCTESWPLAHHRTIYTTFLLLFQYCLPLGFILVCYARIYRR
LQRQGRVFHKGTYSLRAGHMKQVNVVLVVMVVAFAVLWLPLHVFNSLEDWHHEAIPICHG
NLIFLVCHLLAMASTCVNPFIYGFLNTNFKKEIKALVLTCQQSAPLEESEHLPLSTVHTE
VSKGSLRLSGRSNPI
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  Blast E-value cutoff:
BDBM50197025
n/a
NameBDBM50197025
Synonyms:CHEMBL439904 | PYY(3-36)
TypeSmall organic molecule
Emp. Form.C180H279N53O54
Mol. Mass.4049.464
SMILESn/a
Structure
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