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TargetDelta carbonic anhydrase
LigandBDBM26999
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1282543 (CHEMBL3101210)
Ki 169±n/a nM
Citation Vullo, DDel Prete, SOsman, SMDe Luca, VScozzafava, AAlothman, ZSupuran, CTCapasso, C Sulfonamide inhibition studies of thed-carbonic anhydrase from the diatom Thalassiosira weissflogii. Bioorg Med Chem Lett24:275-9 (2013) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Delta carbonic anhydrase
Name:Delta carbonic anhydrase
Synonyms:ca1
Type:PROTEIN
Mol. Mass.:32261.40
Organism:Thalassiosira weissflogii
Description:ChEMBL_107983
Residue:281
Sequence:
MEVDVVPNTKNYWQSSMCPVNVHWHLGTEHYSVGEYDENGSGPNGNVGVPYRRTLAEGEV
QDGFRCHHYDPDDEAYTRPYEWKHCIGMEVGETYEVHWPHSGAGACGTTYQYQTPFYDGV
FCNLDMETLQTLAPQDIANAVGVQGQIFTIVNDDTYYYPDLIRGWIVDEEMGMGQDIAMY
TGSTTGESRSNEICSSYSPITWQVDRKCHKISASSFDKLCYDMKMQRDDMSDDLYAHGSR
ELVTPEYVANNQQTRRLTEKHEHNHSHGHSHVRGHQHHQWF
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM26999
n/a
NameBDBM26999
Synonyms:4-(1,1-dioxo-1,2-thiazinan-2-yl)benzene-1-sulfonamide | CHEMBL328560 | Contravul | Ospolot | Sulthiame (SLT) | Sulthiame, 2
TypeSmall organic molecule
Emp. Form.C10H14N2O4S2
Mol. Mass.290.359
SMILESNS(=O)(=O)c1ccc(cc1)N1CCCCS1(=O)=O
Structure
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