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TargetChromobox protein homolog 7
LigandBDBM50009483
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1336411 (CHEMBL3242415)
IC50 102000±n/a nM
Citation Simhadri, CDaze, KDDouglas, SFQuon, TTDev, AGignac, MCPeng, FHeller, MBoulanger, MJWulff, JEHof, F Chromodomain antagonists that target the polycomb-group methyllysine reader protein chromobox homolog 7 (CBX7). J Med Chem57:2874-83 (2014) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Chromobox protein homolog 7
Name:Chromobox protein homolog 7
Synonyms:CBX7 | CBX7_HUMAN | Chromobox protein homolog 7 | Chromobox protein homolog 7 (CBX7)
Type:Protein
Mol. Mass.:28351.76
Organism:Homo sapiens (Human)
Description:n/a
Residue:251
Sequence:
MELSAIGEQVFAVESIRKKRVRKGKVEYLVKWKGWPPKYSTWEPEEHILDPRLVMAYEEK
EERDRASGYRKRGPKPKRLLLQRLYSMDLRSSHKAKGKEKLCFSLTCPLGSGSPEGVVKA
GAPELVDKGPLVPTLPFPLRKPRKAHKYLRLSRKKFPPRGPNLESHSHRRELFLQEPPAP
DVLQAAGEWEPAAQPPEEEADADLAEGPPPWTPALPSSEVTVTDITANSITVTFREAQAA
EGFFRDRSGKF
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  Blast E-value cutoff:
BDBM50009483
n/a
NameBDBM50009483
Synonyms:CHEMBL3234165
TypeSmall organic molecule
Emp. Form.C32H55N6O5
Mol. Mass.603.8158
SMILESCCCNC(=O)[C@H](CCCC[N+](C)(C)C)NC(=O)[C@H](CC(C)C)NC(=O)[C@H](C)NC(=O)[C@H](Cc1ccccc1)NC(C)=O |r|
Structure
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