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TargetChromobox protein homolog 7
LigandBDBM50009553
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1336412 (CHEMBL3242416)
Kd 220±n/a nM
Citation Simhadri, CDaze, KDDouglas, SFQuon, TTDev, AGignac, MCPeng, FHeller, MBoulanger, MJWulff, JEHof, F Chromodomain antagonists that target the polycomb-group methyllysine reader protein chromobox homolog 7 (CBX7). J Med Chem57:2874-83 (2014) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Chromobox protein homolog 7
Name:Chromobox protein homolog 7
Synonyms:CBX7 | CBX7_HUMAN | Chromobox protein homolog 7 | Chromobox protein homolog 7 (CBX7)
Type:Protein
Mol. Mass.:28351.76
Organism:Homo sapiens (Human)
Description:n/a
Residue:251
Sequence:
MELSAIGEQVFAVESIRKKRVRKGKVEYLVKWKGWPPKYSTWEPEEHILDPRLVMAYEEK
EERDRASGYRKRGPKPKRLLLQRLYSMDLRSSHKAKGKEKLCFSLTCPLGSGSPEGVVKA
GAPELVDKGPLVPTLPFPLRKPRKAHKYLRLSRKKFPPRGPNLESHSHRRELFLQEPPAP
DVLQAAGEWEPAAQPPEEEADADLAEGPPPWTPALPSSEVTVTDITANSITVTFREAQAA
EGFFRDRSGKF
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  Blast E-value cutoff:
BDBM50009553
n/a
NameBDBM50009553
Synonyms:CHEMBL3234441
TypeSmall organic molecule
Emp. Form.C37H56BrN7O5
Mol. Mass.758.787
SMILESC[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)c1ccc(Br)cc1)C(=O)N[C@@H](C1CCCC1)C(=O)N[C@@H](CCCC[N+](C)(C)C)C(=O)NCC[NH3+] |r|
Structure
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