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TargetG-protein coupled receptor 183
LigandBDBM50011701
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1351308
IC50 5.0±n/a nM
Citation Gessier FPreuss IYin HRosenkilde MMLaurent SEndres RChen YAMarsilje THSeuwen KNguyen DGSailer AW Identification and characterization of small molecule modulators of the Epstein-Barr virus-induced gene 2 (EBI2) receptor. J Med Chem 57:3358-68 (2014) [PubMed]  Article
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G-protein coupled receptor 183
Name:G-protein coupled receptor 183
Synonyms:EBI2
Type:PROTEIN
Mol. Mass.:41245.79
Organism:Homo sapiens (Human)
Description:ChEMBL_108311
Residue:361
Sequence:
MDIQMANNFTPPSATPQGNDCDLYAHHSTARIVMPLHYSLVFIIGLVGNLLALVVIVQNR
KKINSTTLYSTNLVISDILFTTALPTRIAYYAMGFDWRIGDALCRITALVFYINTYAGVN
FMTCLSIDRFIAVVHPLRYNKIKRIEHAKGVCIFVWILVFAQTLPLLINPMSKQEAERIT
CMEYPNFEETKSLPWILLGACFIGYVLPLIIILICYSQICCKLFRTAKQNPLTEKSGVNK
KALNTIILIIVVFVLCFTPYHVAIIQHMIKKLRFSNFLECSQRHSFQISLHFTVCLMNFN
CCMDPFIYFFACKGYKRKVMRMLKRQVSVSISSAVKSAPEENSREMTETQMMIHSKSSNG
K
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BDBM50011701
n/a
NameBDBM50011701
Synonyms:CHEMBL3262895
TypeSmall organic molecule
Emp. Form.C22H21BrN2O3
Mol. Mass.441.318
SMILESBrc1ccc(\C=C\C(=O)N2CCN(CC2)C(=O)c2ccc3OCCc3c2)cc1
Structure
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