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TargetG-protein coupled receptor 183
LigandBDBM50011716
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1352280
IC50 7.0±n/a nM
Citation Gessier FPreuss IYin HRosenkilde MMLaurent SEndres RChen YAMarsilje THSeuwen KNguyen DGSailer AW Identification and characterization of small molecule modulators of the Epstein-Barr virus-induced gene 2 (EBI2) receptor. J Med Chem 57:3358-68 (2014) [PubMed]  Article
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G-protein coupled receptor 183
Name:G-protein coupled receptor 183
Synonyms:EBI2
Type:PROTEIN
Mol. Mass.:41245.79
Organism:Homo sapiens (Human)
Description:ChEMBL_108311
Residue:361
Sequence:
MDIQMANNFTPPSATPQGNDCDLYAHHSTARIVMPLHYSLVFIIGLVGNLLALVVIVQNR
KKINSTTLYSTNLVISDILFTTALPTRIAYYAMGFDWRIGDALCRITALVFYINTYAGVN
FMTCLSIDRFIAVVHPLRYNKIKRIEHAKGVCIFVWILVFAQTLPLLINPMSKQEAERIT
CMEYPNFEETKSLPWILLGACFIGYVLPLIIILICYSQICCKLFRTAKQNPLTEKSGVNK
KALNTIILIIVVFVLCFTPYHVAIIQHMIKKLRFSNFLECSQRHSFQISLHFTVCLMNFN
CCMDPFIYFFACKGYKRKVMRMLKRQVSVSISSAVKSAPEENSREMTETQMMIHSKSSNG
K
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  Blast E-value cutoff:
BDBM50011716
n/a
NameBDBM50011716
Synonyms:CHEMBL3262896
TypeSmall organic molecule
Emp. Form.C21H21BrN2O3
Mol. Mass.429.307
SMILESCOc1ccc(cc1)C(=O)N1CCN(CC1)C(=O)\C=C\c1ccc(Br)cc1
Structure
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