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TargetG-protein coupled receptor 183
LigandBDBM50011731
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1351309 (CHEMBL3266158)
IC50 20±n/a nM
Citation Gessier, FPreuss, IYin, HRosenkilde, MMLaurent, SEndres, RChen, YAMarsilje, THSeuwen, KNguyen, DGSailer, AW Identification and characterization of small molecule modulators of the Epstein-Barr virus-induced gene 2 (EBI2) receptor. J Med Chem57:3358-68 (2014) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
G-protein coupled receptor 183
Name:G-protein coupled receptor 183
Synonyms:EBV-induced G-protein coupled receptor 2 | Ebi2 | Epstein-Barr virus-induced G-protein coupled receptor 2 | GP183_MOUSE | Gpr183
Type:PROTEIN
Mol. Mass.:40205.57
Organism:Mus musculus
Description:ChEMBL_108312
Residue:357
Sequence:
MANNFTTPLATSHGNNCDLYAHHSTARVLMPLHYSLVFIIGLVGNLLALVVIVQNRKKIN
STTLYSMNLVISDILFTTALPTRIAYYALGFDWRIGDALCRVTALVFYINTYAGVNFMTC
LSIDRFFAVVHPLRYNKIKRIEYAKGVCLSVWILVFAQTLPLLLTPMSKEEGDKTTCMEY
PNFEGTASLPWILLGACLLGYVLPITVILLCYSQICCKLFRTAKQNPLTEKSGVNKKALN
TIILIIVVFILCFTPYHVAIIQHMIKMLCSPGALECGARHSFQISLHFTVCLMNFNCCMD
PFIYFFACKGYKRKVMKMLKRQVSVSISSAVRSAPEENSREMTESQMMIHSKASNGR
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BDBM50011731
n/a
NameBDBM50011731
Synonyms:CHEMBL3262889
TypeSmall organic molecule
Emp. Form.C23H27N3O3
Mol. Mass.393.4788
SMILESCOc1ccc(\C=C\C(=O)N2CCN(CC2)C(=O)c2ccc(cc2)N(C)C)cc1
Structure
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