| Reaction Details |
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 | Report a problem with these data |
| Target | G-protein coupled receptor 183 |
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| Ligand | BDBM50011578 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1351309 (CHEMBL3266158) |
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| IC50 | 18±n/a nM |
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| Citation |  Gessier, F; Preuss, I; Yin, H; Rosenkilde, MM; Laurent, S; Endres, R; Chen, YA; Marsilje, TH; Seuwen, K; Nguyen, DG; Sailer, AW Identification and characterization of small molecule modulators of the Epstein-Barr virus-induced gene 2 (EBI2) receptor. J Med Chem57:3358-68 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| G-protein coupled receptor 183 |
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| Name: | G-protein coupled receptor 183 |
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| Synonyms: | EBV-induced G-protein coupled receptor 2 | Ebi2 | Epstein-Barr virus-induced G-protein coupled receptor 2 | GP183_MOUSE | Gpr183 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 40205.57 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_108312 |
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| Residue: | 357 |
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| Sequence: | MANNFTTPLATSHGNNCDLYAHHSTARVLMPLHYSLVFIIGLVGNLLALVVIVQNRKKIN
STTLYSMNLVISDILFTTALPTRIAYYALGFDWRIGDALCRVTALVFYINTYAGVNFMTC
LSIDRFFAVVHPLRYNKIKRIEYAKGVCLSVWILVFAQTLPLLLTPMSKEEGDKTTCMEY
PNFEGTASLPWILLGACLLGYVLPITVILLCYSQICCKLFRTAKQNPLTEKSGVNKKALN
TIILIIVVFILCFTPYHVAIIQHMIKMLCSPGALECGARHSFQISLHFTVCLMNFNCCMD
PFIYFFACKGYKRKVMKMLKRQVSVSISSAVRSAPEENSREMTESQMMIHSKASNGR
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| BDBM50011578 |
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| n/a |
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| Name | BDBM50011578 |
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| Synonyms: | CHEMBL3262890 |
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| Type | Small organic molecule |
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| Emp. Form. | C23H24N2O5 |
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| Mol. Mass. | 408.4471 |
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| SMILES | COC(=O)c1ccc(cc1)C(=O)N1CCN(CC1)C(=O)\C=C\c1ccc(OC)cc1 |
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| Structure | 
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