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TargetG-protein coupled receptor 183
LigandBDBM50011701
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1351309
IC50 6.0±n/a nM
Citation Gessier FPreuss IYin HRosenkilde MMLaurent SEndres RChen YAMarsilje THSeuwen KNguyen DGSailer AW Identification and characterization of small molecule modulators of the Epstein-Barr virus-induced gene 2 (EBI2) receptor. J Med Chem 57:3358-68 (2014) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
G-protein coupled receptor 183
Name:G-protein coupled receptor 183
Synonyms:EBI2 | EBV-induced G-protein coupled receptor 2 | Ebi2 | Epstein-Barr virus-induced G-protein coupled receptor 2 | Gpr183
Type:PROTEIN
Mol. Mass.:40205.57
Organism:Mus musculus
Description:ChEMBL_108312
Residue:357
Sequence:
MANNFTTPLATSHGNNCDLYAHHSTARVLMPLHYSLVFIIGLVGNLLALVVIVQNRKKIN
STTLYSMNLVISDILFTTALPTRIAYYALGFDWRIGDALCRVTALVFYINTYAGVNFMTC
LSIDRFFAVVHPLRYNKIKRIEYAKGVCLSVWILVFAQTLPLLLTPMSKEEGDKTTCMEY
PNFEGTASLPWILLGACLLGYVLPITVILLCYSQICCKLFRTAKQNPLTEKSGVNKKALN
TIILIIVVFILCFTPYHVAIIQHMIKMLCSPGALECGARHSFQISLHFTVCLMNFNCCMD
PFIYFFACKGYKRKVMKMLKRQVSVSISSAVRSAPEENSREMTESQMMIHSKASNGR
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  Blast E-value cutoff:
BDBM50011701
n/a
NameBDBM50011701
Synonyms:CHEMBL3262895
TypeSmall organic molecule
Emp. Form.C22H21BrN2O3
Mol. Mass.441.318
SMILESBrc1ccc(\C=C\C(=O)N2CCN(CC2)C(=O)c2ccc3OCCc3c2)cc1
Structure
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