| Reaction Details |
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 | Report a problem with these data |
| Target | Arylamine N-acetyltransferase 2 |
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| Ligand | BDBM50014986 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1347887 (CHEMBL3267123) |
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| IC50 | 270±n/a nM |
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| Citation |  Egleton, JE; Thinnes, CC; Seden, PT; Laurieri, N; Lee, SP; Hadavizadeh, KS; Measures, AR; Jones, AM; Thompson, S; Varney, A; Wynne, GM; Ryan, A; Sim, E; Russell, AJ Structure-activity relationships and colorimetric properties of specific probes for the putative cancer biomarker human arylamine N-acetyltransferase 1. Bioorg Med Chem22:3030-54 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Arylamine N-acetyltransferase 2 |
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| Name: | Arylamine N-acetyltransferase 2 |
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| Synonyms: | ARY2_MOUSE | Aac2 | Nat2 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 33697.98 |
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| Organism: | Mus musculus |
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| Description: | ChEMBL_1347887 |
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| Residue: | 290 |
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| Sequence: | MDIEAYFERIGYQSTRSKLDLKTLTEILQHQIRAIPFENLNIHCGESMELSLEAIFDQIV
RKKRGGWCLQVNHLLYWALTKLGFETTMLGGYVFNTPANKYSSGMIHLLVQVTISGKDYI
VDAGFGRSYQMWEPLELTSGKDQPQVPAIFRLTEENGTWYLDQIRREQYVPNQEFINSDL
LEKNKYRKIYSFTLEPRTIEDFESMNTYLQTSPASVFTSKSFCSLQTPEGVHCLVGSTLT
YRRFSYKDNVDLVEFKSLTEEEIEDVLRTIFGVSLERKLVPKHGDRFFTI
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| BDBM50014986 |
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| n/a |
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| Name | BDBM50014986 |
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| Synonyms: | CHEMBL3262086 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H17N3O4S |
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| Mol. Mass. | 419.453 |
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| SMILES | Nc1cccc2C(=O)C(Nc3ccccc3)=C(NS(=O)(=O)c3ccccc3)C(=O)c12 |t:16| |
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| Structure | 
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