Reaction Details |
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Target | Glandular kallikrein |
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Ligand | BDBM50016544 |
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Substrate/Competitor | n/a |
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Meas. Tech. | ChEMBL_1354676 (CHEMBL3281101) |
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Ki | 1600±n/a nM |
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Citation | Geratz, JD; Cheng, MC; Tidwell, RR Novel bis(benzamidino) compounds with an aromatic central link. Inhibitors of thrombin, pancreatic kallikrein, trypsin, and complement. J Med Chem19:634-9 (1976) [PubMed] |
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More Info.: | Get all data from this article, Assay Method |
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Glandular kallikrein |
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Name: | Glandular kallikrein |
Synonyms: | KLK_PIG | Tissue kallikrein |
Type: | PROTEIN |
Mol. Mass.: | 26710.38 |
Organism: | Sus scrofa |
Description: | ChEMBL_108296 |
Residue: | 242 |
Sequence: | APPIQSRIIGGRECEKNSHPWQVAIYHYSSFQCGGVLVNPKWVLTAAHCKNDNYEVWLGR
HNLFENENTAQFFGVTADFPHPGFNLSLLKHTKADGKDYSHDLMLLRLQSPAKITDAVKV
LELPTQEPELGSTCEASGWGSIEPGPDFEFPDEIQCVQLTLLQNTFCAAHPKVTESMLCA
GYLPGGKDTCMGDSGGPLICNGMWQGITSWGHTPCGSANKPSIYTKLIFYLDWINDTITE
NP
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BDBM50016544 |
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n/a |
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Name | BDBM50016544 |
Synonyms: | CHEMBL3277934 |
Type | Small organic molecule |
Emp. Form. | C28H27ClN4O2 |
Mol. Mass. | 486.993 |
SMILES | Cl.NC(=N)c1ccc(OCc2cccc(c2)-c2cccc(COc3ccc(cc3)C(N)=N)c2)cc1 |
Structure |
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