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TargetGlandular kallikrein
LigandBDBM50016544
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1354676 (CHEMBL3281101)
Ki 1600±n/a nM
Citation Geratz, JDCheng, MCTidwell, RR Novel bis(benzamidino) compounds with an aromatic central link. Inhibitors of thrombin, pancreatic kallikrein, trypsin, and complement. J Med Chem19:634-9 (1976) [PubMed]
More Info.:Get all data from this article,  Assay Method
 
Glandular kallikrein
Name:Glandular kallikrein
Synonyms:KLK_PIG | Tissue kallikrein
Type:PROTEIN
Mol. Mass.:26710.38
Organism:Sus scrofa
Description:ChEMBL_108296
Residue:242
Sequence:
APPIQSRIIGGRECEKNSHPWQVAIYHYSSFQCGGVLVNPKWVLTAAHCKNDNYEVWLGR
HNLFENENTAQFFGVTADFPHPGFNLSLLKHTKADGKDYSHDLMLLRLQSPAKITDAVKV
LELPTQEPELGSTCEASGWGSIEPGPDFEFPDEIQCVQLTLLQNTFCAAHPKVTESMLCA
GYLPGGKDTCMGDSGGPLICNGMWQGITSWGHTPCGSANKPSIYTKLIFYLDWINDTITE
NP
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BDBM50016544
n/a
NameBDBM50016544
Synonyms:CHEMBL3277934
TypeSmall organic molecule
Emp. Form.C28H27ClN4O2
Mol. Mass.486.993
SMILESCl.NC(=N)c1ccc(OCc2cccc(c2)-c2cccc(COc3ccc(cc3)C(N)=N)c2)cc1
Structure
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