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TargetMatrix protein 2
LigandBDBM50020844
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1364624 (CHEMBL3291757)
IC50 4930±n/a nM
Citation Rey-Carrizo, MBarniol-Xicota, MMa, CFrigolé-Vivas, MTorres, ENaesens, LLlabrés, SJuárez-Jiménez, JLuque, FJDeGrado, WFLamb, RAPinto, LHVázquez, S Easily accessible polycyclic amines that inhibit the wild-type and amantadine-resistant mutants of the M2 channel of influenza A virus. J Med Chem57:5738-47 (2014) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Matrix protein 2
Name:Matrix protein 2
Synonyms:M | M2_I72A8 | Proton channel protein M2
Type:PROTEIN
Mol. Mass.:11180.06
Organism:Influenza A virus (A/Udorn/307/1972(H3N2))
Description:ChEMBL_22
Residue:97
Sequence:
MSLLTEVETPIRNEWGCRCNDSSDPLVVAASIIGILHLILWILDRLFFKCIYRFFEHGLK
RGPSTEGVPESMREEYRKEQQSAVDADDSHFVSIELE
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BDBM50020844
n/a
NameBDBM50020844
Synonyms:CHEMBL3286403
TypeSmall organic molecule
Emp. Form.C13H18ClN3
Mol. Mass.251.755
SMILESCl.NC(=N)N1CC2C(C1)C1C=CC2C2C=CC12 |c:10,15,TLB:5:6:10.11:13.16,THB:8:7:10.11:13.16,15:16:10.11:7.6,14:13:10.11:7.6|
Structure
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