| Reaction Details |
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 | Report a problem with these data |
| Target | Somatostatin receptor type 2 |
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| Ligand | BDBM50021063 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1365879 (CHEMBL3296537) |
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| Ki | 311±n/a nM |
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| Citation |  Li, D; Wu, Z; Yu, Y; Ball, RG; Guo, L; Sherer, E; He, S; Hong, Q; Lai, Z; Qi, H; Truong, Q; Yang, DX; Chicchi, GG; Tsao, KL; Trusca, D; Trujillo, M; Pachanski, M; Eiermann, GJ; Howard, AD; Zhou, YP; Zhang, BB; Nargund, RP; Hagmann, WK Diamine Derivatives as Novel Small-Molecule, Potent, and Subtype-Selective Somatostatin SST3 Receptor Agonists. ACS Med Chem Lett5:690-5 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Somatostatin receptor type 2 |
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| Name: | Somatostatin receptor type 2 |
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| Synonyms: | SOMATOSTATIN SST2 | SRIF-1 | SS-2-R | SS2-R | SS2R | SSR2_HUMAN | SSTR2 | Somatostatin receptor type 2 (SSTR2) |
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| Type: | Enzyme |
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| Mol. Mass.: | 41344.94 |
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| Organism: | Homo sapiens (Human) |
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| Description: | P30874 |
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| Residue: | 369 |
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| Sequence: | MDMADEPLNGSHTWLSIPFDLNGSVVSTNTSNQTEPYYDLTSNAVLTFIYFVVCIIGLCG
NTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMT
VDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMITMAVWGVSLLVILPIMIY
AGLRSNQWGRSSCTINWPGESGAWYTGFIIYTFILGFLVPLTIICLCYLFIIIKVKSSGI
RVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSMAISPTPALKGMFDFVVVL
TYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGTDDGERSDSKQDKSRLNETTETQRTL
LNGDLQTSI
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| BDBM50021063 |
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| n/a |
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| Name | BDBM50021063 |
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| Synonyms: | CHEMBL3287613 |
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| Type | Small organic molecule |
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| Emp. Form. | C22H24FN3O |
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| Mol. Mass. | 365.4439 |
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| SMILES | Fc1ccc(cc1)C(=O)N[C@@H]1CCCC[C@@H]1NCc1c[nH]c2ccccc12 |r| |
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| Structure | 
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