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TargetLeucine aminopeptidase (LAP)
LigandBDBM50024597
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1442056
Ki 220±n/a nM
Citation Vassiliou SWeglarz-Tomczak EBerlicki LPawelczak MNocek BMulligan RJoachimiak AMucha A Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases. J Med Chem 57:8140-51 (2014) [PubMed]  Article
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Leucine aminopeptidase (LAP)
Name:Leucine aminopeptidase (LAP)
Synonyms:Cytosol aminopeptidase
Type:Enzyme
Mol. Mass.:4015.44
Organism:Sus scrofa (Pig)
Description:P28839
Residue:36
Sequence:
TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
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  Blast E-value cutoff:
BDBM50024597
n/a
NameBDBM50024597
Synonyms:(S)-1-Ammonium-3-methyl-butane-1-phosphonic acid anion | CHEMBL288165
TypeSmall organic molecule
Emp. Form.C5H14NO3P
Mol. Mass.167.1433
SMILESCC(C)C[C@@H]([NH3+])P(O)([O-])=O
Structure
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