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TargetCytosol aminopeptidase [33-68,L62W]
LigandBDBM50024597
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1442056 (CHEMBL3373424)
Ki 220±n/a nM
Citation Vassiliou, SWeglarz-Tomczak, EBerlicki, LPawelczak, MNocek, BMulligan, RJoachimiak, AMucha, A Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases. J Med Chem57:8140-51 (2014) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Cytosol aminopeptidase [33-68,L62W]
Name:Cytosol aminopeptidase [33-68,L62W]
Synonyms:AMPL_PIG | Cytosol aminopeptidase | LAP3 | Leucine aminopeptidase (LAP)
Type:Enzyme
Mol. Mass.:4015.44
Organism:Sus scrofa (Pig)
Description:P28839[33-68,L62W]
Residue:36
Sequence:
TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
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  Blast E-value cutoff:
BDBM50024597
n/a
NameBDBM50024597
Synonyms:(S)-1-Ammonium-3-methyl-butane-1-phosphonic acid anion | CHEMBL288165
TypeSmall organic molecule
Emp. Form.C5H14NO3P
Mol. Mass.167.1433
SMILESCC(C)C[C@@H]([NH3+])P(O)([O-])=O
Structure
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