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TargetLeucine aminopeptidase (LAP)
LigandBDBM50078125
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1442056
Ki 7.7±n/a nM
Citation Vassiliou SWeglarz-Tomczak EBerlicki LPawelczak MNocek BMulligan RJoachimiak AMucha A Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases. J Med Chem 57:8140-51 (2014) [PubMed]  Article
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Leucine aminopeptidase (LAP)
Name:Leucine aminopeptidase (LAP)
Synonyms:Cytosol aminopeptidase
Type:Enzyme
Mol. Mass.:4015.44
Organism:Sus scrofa (Pig)
Description:P28839
Residue:36
Sequence:
TKGLVLGIYSKEKEDDAPQFTSAGENFDKWVSGKLR
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  Blast E-value cutoff:
BDBM50078125
n/a
NameBDBM50078125
Synonyms:(1-Amino-3-phenyl-propyl)-phosphinic acid | CHEMBL289824
TypeSmall organic molecule
Emp. Form.C9H12NO2P
Mol. Mass.197.1708
SMILESOP(O)C(=N)CCc1ccccc1
Structure
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