| Reaction Details |
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 | Report a problem with these data |
| Target | Mu-type opioid receptor |
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| Ligand | BDBM50028085 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1434014 (CHEMBL3381486) |
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| Ki | >1000±n/a nM |
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| Citation |  Hirayama, S; Wada, N; Kuroda, N; Iwai, T; Yamaotsu, N; Hirono, S; Fujii, H; Nagase, H Synthesis of a novel universal opioid receptor agonist with the 1,3,5-trioxazatriquinane skeleton and its pharmacologies. Bioorg Med Chem Lett24:4895-8 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Mu-type opioid receptor |
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| Name: | Mu-type opioid receptor |
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| Synonyms: | M-OR-1 | MOR-1 | Mor | OPIATE Mu | OPRM_MOUSE | Opioid receptors; mu and delta | Oprm | Oprm1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 44431.62 |
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| Organism: | MOUSE |
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| Description: | OPIATE Mu OPRM1 MOUSE::P42866 |
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| Residue: | 398 |
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| Sequence: | MDSSAGPGNISDCSDPLAPASCSPAPGSWLNLSHVDGNQSDPCGPNRTGLGGSHSLCPQT
GSPSMVTAITIMALYSIVCVVGLFGNFLVMYVIVRYTKMKTATNIYIFNLALADALATST
LPFQSVNYLMGTWPFGNILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRT
PRNAKIVNVCNWILSSAIGLPVMFMATTKYRQGSIDCTLTFSHPTWYWENLLKICVFIFA
FIMPVLIITVCYGLMILRLKSVRMLSGSKEKDRNLRRITRMVLVVVAVFIVCWTPIHIYV
IIKALITIPETTFQTVSWHFCIALGYTNSCLNPVLYAFLDENFKRCFREFCIPTSSTIEQ
QNSARIRQNTREHPSTANTVDRTNHQLENLEAETAPLP
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| BDBM50028085 |
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| n/a |
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| Name | BDBM50028085 |
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| Synonyms: | CHEMBL3338871 |
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| Type | Small organic molecule |
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| Emp. Form. | C27H27NO6 |
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| Mol. Mass. | 461.5064 |
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| SMILES | [H][C@]12O[C@@](C)(c3ccc(O)cc3)[C@]3([H])O[C@@](C)(c4ccc(O)cc4)[C@]([H])(O[C@]1(C)c1ccc(O)cc1)N23 |r| |
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| Structure | 
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