| Reaction Details |
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 | Report a problem with these data |
| Target | Delta-type opioid receptor |
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| Ligand | BDBM50028087 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1434015 (CHEMBL3381487) |
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| Ki | >1000±n/a nM |
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| Citation |  Hirayama, S; Wada, N; Kuroda, N; Iwai, T; Yamaotsu, N; Hirono, S; Fujii, H; Nagase, H Synthesis of a novel universal opioid receptor agonist with the 1,3,5-trioxazatriquinane skeleton and its pharmacologies. Bioorg Med Chem Lett24:4895-8 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Delta-type opioid receptor |
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| Name: | Delta-type opioid receptor |
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| Synonyms: | DOR-1 | K56 | MSL-2 | OPIATE Delta | OPRD_MOUSE | Opioid receptors; mu and delta | Oprd1 |
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| Type: | Enzyme Catalytic Domain |
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| Mol. Mass.: | 40577.25 |
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| Organism: | MOUSE |
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| Description: | P32300 |
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| Residue: | 372 |
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| Sequence: | MELVPSARAELQSSPLVNLSDAFPSAFPSAGANASGSPGARSASSLALAIAITALYSAVC
AVGLLGNVLVMFGIVRYTKLKTATNIYIFNLALADALATSTLPFQSAKYLMETWPFGELL
CKAVLSIDYYNMFTSIFTLTMMSVDRYIAVCHPVKALDFRTPAKAKLINICIWVLASGVG
VPIMVMAVTQPRDGAVVCMLQFPSPSWYWDTVTKICVFLFAFVVPILIITVCYGLMLLRL
RSVRLLSGSKEKDRSLRRITRMVLVVVGAFVVCWAPIHIFVIVWTLVDINRRDPLVVAAL
HLCIALGYANSSLNPVLYAFLDENFKRCFRQLCRTPCGRQEPGSLRRPRQATTRERVTAC
TPSDGPGGGAAA
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| BDBM50028087 |
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| n/a |
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| Name | BDBM50028087 |
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| Synonyms: | CHEMBL3338884 |
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| Type | Small organic molecule |
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| Emp. Form. | C13H15NO4 |
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| Mol. Mass. | 249.2625 |
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| SMILES | [H][C@]12CO[C@]3([H])N1[C@]([H])(CO2)O[C@]3(C)c1ccc(O)cc1 |r| |
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| Structure | 
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