| Reaction Details |
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 | Report a problem with these data |
| Target | Neuropeptide FF receptor 1 |
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| Ligand | BDBM50029185 |
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| Substrate/Competitor | n/a |
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| Meas. Tech. | ChEMBL_1436237 (CHEMBL3387184) |
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| Ki | 479±n/a nM |
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| Citation |  Journigan, VB; Mésangeau, C; Vyas, N; Eans, SO; Cutler, SJ; McLaughlin, JP; Mollereau, C; McCurdy, CR Nonpeptide small molecule agonist and antagonist original leads for neuropeptide FF1 and FF2 receptors. J Med Chem57:8903-27 (2014) [PubMed] Article |
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| More Info.: | Get all data from this article, Assay Method |
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| Neuropeptide FF receptor 1 |
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| Name: | Neuropeptide FF receptor 1 |
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| Synonyms: | G-protein coupled receptor 147 | GPR147 | NPFF1 | NPFF1_HUMAN | NPFFR1 | RFamide-related peptide receptor OT7T022 |
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| Type: | PROTEIN |
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| Mol. Mass.: | 47840.07 |
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| Organism: | Homo sapiens (Human) |
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| Description: | ChEMBL_1474637 |
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| Residue: | 430 |
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| Sequence: | MEGEPSQPPNSSWPLSQNGTNTEATPATNLTFSSYYQHTSPVAAMFIVAYALIFLLCMVG
NTLVCFIVLKNRHMHTVTNMFILNLAVSDLLVGIFCMPTTLVDNLITGWPFDNATCKMSG
LVQGMSVSASVFTLVAIAVERFRCIVHPFREKLTLRKALVTIAVIWALALLIMCPSAVTL
TVTREEHHFMVDARNRSYPLYSCWEAWPEKGMRRVYTTVLFSHIYLAPLALIVVMYARIA
RKLCQAPGPAPGGEEAADPRASRRRARVVHMLVMVALFFTLSWLPLWALLLLIDYGQLSA
PQLHLVTVYAFPFAHWLAFFNSSANPIIYGYFNENFRRGFQAAFRARLCPRPSGSHKEAY
SERPGGLLHRRVFVVVRPSDSGLPSESGPSSGAPRPGRLPLRNGRVAHHGLPREGPGCSH
LPLTIPAWDI
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| BDBM50029185 |
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| n/a |
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| Name | BDBM50029185 |
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| Synonyms: | CHEMBL3360834 |
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| Type | Small organic molecule |
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| Emp. Form. | C29H39N7O |
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| Mol. Mass. | 501.6663 |
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| SMILES | N[C@@H](CCCNC(N)=N)C(=O)NCC1(CCN(Cc2ccc3ccccc3c2)CC1)Nc1ccccc1 |r| |
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| Structure | 
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