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TargetProtein delta homolog 1
LigandBDBM50042940
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1444684
Ki 0.400000±n/a nM
Citation Abdel-Magid AF Dual leucine zipper kinase inhibitors: potential treatments for neurodegenerative diseases. ACS Med Chem Lett 6:11-2 (2015) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Protein delta homolog 1
Name:Protein delta homolog 1
Synonyms:DLK-1 | FA1 | Fetal antigen 1 | pG2
Type:PROTEIN
Mol. Mass.:41294.81
Organism:Homo sapiens (Human)
Description:ChEMBL_1444684
Residue:383
Sequence:
MTATEALLRVLLLLLAFGHSTYGAECFPACNPQNGFCEDDNVCRCQPGWQGPLCDQCVTS
PGCLHGLCGEPGQCICTDGWDGELCDRDVRACSSAPCANNRTCVSLDDGLYECSCAPGYS
GKDCQKKDGPCVINGSPCQHGGTCVDDEGRASHASCLCPPGFSGNFCEIVANSCTPNPCE
NDGVCTDIGGDFRCRCPAGFIDKTCSRPVTNCASSPCQNGGTCLQHTQVSYECLCKPEFT
GLTCVKKRALSPQQVTRLPSGYGLAYRLTPGVHELPVQQPEHRILKVSMKELNKKTPLLT
EGQAICFTILGVLTSLVVLGTVGIVFLNKCETWVSNLRYNHMLRKKKNLLLQYNSGEDLA
VNIIFPEKIDMTTFSKEAGDEEI
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50042940
n/a
NameBDBM50042940
Synonyms:CHEMBL3355005
TypeSmall organic molecule
Emp. Form.C22H24F3N5O
Mol. Mass.431.4541
SMILES[H][C@@]12CN(C[C@]1([H])[C@H]2c1cc(nn1C(C)C)-c1cnc2[nH]cc(c2c1)C(F)(F)F)C1COC1 |r|
Structure
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