| Reaction Details |
|---|
 | Report a problem with these data |
| Target | Somatostatin receptor type 4 |
|---|
| Ligand | BDBM50445614 |
|---|
| Substrate/Competitor | n/a |
|---|
| Meas. Tech. | ChEMBL_1450033 (CHEMBL3373295) |
|---|
| Ki | >10000±n/a nM |
|---|
| Citation |  Rajagopalan, P; Tracey, H; Chen, Z; Bandyopadhyaya, A; Veeraraghavan, S; Rajagopalan, DR; Salvemini, D; McPhee, I; Viswanadha, S; Rajagopalan, R DDD-028: a potent potential non-opioid, non-cannabinoid analgesic for neuropathic and inflammatory pain. Bioorg Med Chem Lett24:3088-91 (2014) [PubMed] Article |
|---|
| More Info.: | Get all data from this article, Assay Method |
|---|
| |
| Somatostatin receptor type 4 |
|---|
| Name: | Somatostatin receptor type 4 |
|---|
| Synonyms: | SOMATOSTATIN SST4 | SS-4-R | SS4-R | SS4R | SSR4_HUMAN | SST4R | SSTR4 | Somatostatin receptor type 4 (SSTR4) |
|---|
| Type: | Enzyme |
|---|
| Mol. Mass.: | 42015.38 |
|---|
| Organism: | Homo sapiens (Human) |
|---|
| Description: | P31391 |
|---|
| Residue: | 388 |
|---|
| Sequence: | MSAPSTLPPGGEEGLGTAWPSAANASSAPAEAEEAVAGPGDARAAGMVAIQCIYALVCLV
GLVGNALVIFVILRYAKMKTATNIYLLNLAVADELFMLSVPFVASSAALRHWPFGSVLCR
AVLSVDGLNMFTSVFCLTVLSVDRYVAVVHPLRAATYRRPSVAKLINLGVWLASLLVTLP
IAIFADTRPARGGQAVACNLQWPHPAWSAVFVVYTFLLGFLLPVLAIGLCYLLIVGKMRA
VALRAGWQQRRRSEKKITRLVLMVVVVFVLCWMPFYVVQLLNLFVTSLDATVNHVSLILS
YANSCANPILYGFLSDNFRRFFQRVLCLRCCLLEGAGGAEEEPLDYYATALKSKGGAGCM
CPPLPCQQEALQPEPGRKRIPLTRTTTF
|
|
|
|---|
| BDBM50445614 |
|---|
| n/a |
|---|
| Name | BDBM50445614 |
|---|
| Synonyms: | CHEMBL3104093 |
|---|
| Type | Small organic molecule |
|---|
| Emp. Form. | C20H20N2 |
|---|
| Mol. Mass. | 288.3862 |
|---|
| SMILES | CN1CCc2c(C1)c1cccc3-c4ccccc4CCn2c13 |
|---|
| Structure | 
|
|---|
Search and Browse
