Ki Summary BindingDB logo
myBDB logout
Reaction Details
Report a problem with these data
TargetFree fatty acid receptor 4
LigandBDBM50044849
Substrate/Competitorn/a
Meas. Tech.ChEMBL_1455264 (CHEMBL3362270)
EC50 6310±n/a nM
Citation Sparks, SMChen, GCollins, JLDanger, DDock, STJayawickreme, CJenkinson, SLaudeman, CLeesnitzer, MALiang, XMaloney, PMcCoy, DCMoncol, DRash, VRimele, TVulimiri, PWay, JMRoss, S Identification of diarylsulfonamides as agonists of the free fatty acid receptor 4 (FFA4/GPR120). Bioorg Med Chem Lett24:3100-3 (2014) [PubMed]  Article
More Info.:Get all data from this article,  Assay Method
 
Free fatty acid receptor 4
Name:Free fatty acid receptor 4
Synonyms:FFAR4_MOUSE | Ffar4 | Free fatty acid receptor 4 | G-protein coupled receptor GT01 | Gpr120 | O3far1 | Omega-3 fatty acid receptor 1
Type:PROTEIN
Mol. Mass.:40828.60
Organism:Mus musculus
Description:ChEMBL_1454435
Residue:361
Sequence:
MSPECAQTTGPGPSHTLDQVNRTHFPFFSDVKGDHRLVLSVVETTVLGLIFVVSLLGNVC
ALVLVARRRRRGATASLVLNLFCADLLFTSAIPLVLVVRWTEAWLLGPVVCHLLFYVMTM
SGSVTILTLAAVSLERMVCIVRLRRGLSGPGRRTQAALLAFIWGYSALAALPLCILFRVV
PQRLPGGDQEIPICTLDWPNRIGEISWDVFFVTLNFLVPGLVIVISYSKILQITKASRKR
LTLSLAYSESHQIRVSQQDYRLFRTLFLLMVSFFIMWSPIIITILLILIQNFRQDLVIWP
SLFFWVVAFTFANSALNPILYNMSLFRNEWRKIFCCFFFPEKGAIFTDTSVRRNDLSVIS
S
Blast this sequence in BindingDB or PDB
  Blast E-value cutoff:
BDBM50044849
n/a
NameBDBM50044849
Synonyms:CHEMBL3311308
TypeSmall organic molecule
Emp. Form.C16H19NO3S
Mol. Mass.305.392
SMILESCOc1ccc(cc1)S(=O)(=O)Nc1c(C)cc(C)cc1C
Structure
Search PDB for entries with ligand similarity:Similarity to this molecule at least: